CABERGOLINE 20 tabs 0,25mg/tab ZPHC
Cabergoline 0.25 mg/tab. Pack: 20 tablets (1 blister). Manufacturer: ZPHC, Kitay.
Description
Cabergoline — is agonist dofaminovykh receptors, derivative ergolina, primenyaemoe for reduction level prolaktina in krovi. On deystvuet in pituitary, podavlyaya secretion prolaktina and normalizuya gormonalnyy fon. Ispolzuetsya in meditsinskoy praktike in giperprolaktinemii, a also in gormonalnykh skhemakh for kontrolya adverse effects, vyzvannykh increasem prolaktina. The product obladaet prolongirovannym deystviem and sokhranyaet effekt do 7–10 days after intake.
Specifications
• Drug class – prolactin inhibitor;
• Chemical formula – C26H37N5O2;
• Administration – oral;
• Mechanism of action – blokirovka sekretsii prolaktina;
• Half-life ≈ 2-3 day;
• Complete action ≈ do 5 days;
• Dosage ≈ from 0.5 do 1 mg raz in 4-5 days;
• Reduction blood blood pressure – moderate (dose-dependent);
• Head bol – moderate (dose-dependent);
• Reduction synthesis testosterone – net;
• Gepatotoksichnost – possible (mild).
Composition / properties
Dosage form: tablets
Quantity: 20 tablets
Dosage: 0.25 mg per tablet
Active ingredient: Cabergoline
Manufacturer: ZPHC
Country of origin: Kitay
Category: dofaminergicheskie agonisty (ingibitory prolaktina)
Product FAQ
Main effects
● Reduction level prolaktina.
● Vosstanovlenie libido and potentsii.
● Reduction riska gynecomastia, svyazannoy with prolaktinom.
● Improved overall well-being and tone.
● Normalizatsiya level dofamina. --- [Q] Who it is suitable for
● for men with povyshennym prolaktinom (po analizam).
● Polzovatelyam, u kotorykh nablyudayutsya simptomy giperprolaktinemii.
● for those, kto prokhodit gormonalnuyu terapiyu and nuzhdaetsya in kontrole prolaktina. --- [Q] Pharmacokinetics
● Vremya action: do 10 days.
● Period elimination: 63–69 hours.
● Maksimalnaya kontsentratsiya dostigaetsya every 2–3 chasa after intake.
● Metaboliziruetsya in liver, vyvoditsya with kalom and mochoy.
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